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中国科学院海洋研究所机构知识库
Knowledge Management System Of Institute of Oceanology, Chinese Academy of Sciences
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An UHPLC-TOF-MS method for quantifying novel brominated anticancer compound bromophenol-thiosemicarbazone hybrid and its application to in vivo pharmacokinetic study
期刊论文
JOURNAL OF ANALYTICAL SCIENCE AND TECHNOLOGY, 2020, 卷号: 11, 期号: 1, 页码: 7
Authors:
Li, Xiuxue
;
Wang, Lijun
;
Jia, Xiaoling
;
Guo, Chuanlong
;
Li, Chao
;
Zhang, Jiajia
;
Shi, Dayong
Adobe PDF(579Kb)
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View/Download:2/0
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Submit date:2020/09/23
Novel compound
Quantitation
UHPLC-TOF-MS
Pharmacokinetics
Design, synthesis and biological evaluation of bromophenol-thiazolylhydrazone hybrids inhibiting the interaction of translation initiation factors eIF4E/eIF4G as multifunctional agents for cancer treatment
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 177, 页码: 153-170
Authors:
Wang, Lijun
;
Guo, Chuanlong
;
Li, Xiuxue
;
Yu, Xuemin
;
Li, Xiangqian
;
Xu, Kuo
;
Jiang, Bo
;
Jia, Xiaoling
;
Li, Chao
;
Shi, Dayong
Adobe PDF(4835Kb)
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Submit date:2019/08/29
Bromophenol-thiazolylhydrazone hybrids
Synthesis
Multifunctional agents
eIF4E/eIF4G interaction
Autophagy
ROS
Highly Selective Protein Tyrosine Phosphatase Inhibitor, 2,2 ',3,3 '-Tetrabromo-4,4 ',5,5 '-tetrahydroxydiphenylmethane, Ameliorates Type 2 Diabetes Mellitus in BKS db Mice
期刊论文
MOLECULAR PHARMACEUTICS, 2019, 卷号: 16, 期号: 5, 页码: 1839-1850
Authors:
Li, Chao
;
Luo, Jiao
;
Guo, Shuju
;
Jia, Xiaoling
;
Guo, Chuanlong
;
Li, Xiangqian
;
Xu, Qi
;
Shi, Dayong
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Submit date:2019/08/28
type 2 diabetes mellitus
protein tyrosine phosphatase 1B
insulin resistance
hypoglycemic activity
dyslipidemia
CYC27 Synthetic Derivative of Bromophenol from Red Alga Rhodomela confervoides: Anti-Diabetic Effects of Sensitizing Insulin Signaling Pathways and Modulating RNA Splicing-Associated RBPs
期刊论文
MARINE DRUGS, 2019, 卷号: 17, 期号: 1, 页码: 15
Authors:
Luo, Jiao
;
Jiang, Bo
;
Li, Chao
;
Jia, Xiaoling
;
Shi, Dayong
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Submit date:2019/08/28
brominated organic compounds
hypoglycemic activity
insulin-sensitizing effect
RBPs
RNA splicing
Phytochemical and chemotaxonomic study on Leathesia nana (Chordariaceae)
期刊论文
BIOCHEMICAL SYSTEMATICS AND ECOLOGY, 2018, 卷号: 81, 页码: 42-44
Authors:
Xu, Kuo
;
Guo, Shuju
;
Jia, Xiaoling
;
Li, Xiang
;
Shi, Dayong
Adobe PDF(298Kb)
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View/Download:33/0
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Submit date:2019/05/15
Leathesia nana
Chordariaceae
Bromophenol
Chemotaxonomy
PTP1B
Selectivity, cell permeability and oral availability studies of novel bromophenol derivative HPN as protein tyrosine phosphatase 1B inhibitor
期刊论文
BRITISH JOURNAL OF PHARMACOLOGY, 2018, 卷号: 175, 期号: 1, 页码: 140-153
Authors:
Luo, Jiao
;
Xu, Qi
;
Jiang, Bo
;
Zhang, Renshuai
;
Jia, Xiaoling
;
Li, Xiangqian
;
Wang, Lijun
;
Guo, Chuanlong
;
Wu, Ning
;
Shi, Dayong
Adobe PDF(2211Kb)
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View/Download:28/0
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Submit date:2019/08/20