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Discovery of 5-(3-bromo-2-(2,3-dibromo-4,5-dimethoxybenzyl)-4,5-dimethoxybenzylidene)thiazolidine-2,4-dione as a novel potent protein tyrosine phosphatase 1B inhibitor with antidiabetic properties 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 108, 页码: 13
作者:  Jiang, Bo;  Luo, Jiao;  Guo, Shuju;  Wang, Lijun
Adobe PDF(8153Kb)  |  收藏  |  浏览/下载:192/0  |  提交时间:2021/05/11
Type 2 diabetes mellitus  Protein tyrosine phosphatase 1B inhibitors  Thiazolidinedione  Insulin signaling  Anti-diabetic activities  
Design, synthesis and biological evaluation of novel pyrimidinedione derivatives as DPP-4 inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 12, 页码: 2131-2135
作者:  Li, Ning;  Wang, Li-Jun;  Jiang, Bo;  Guo, Shu-Ju;  Li, Xiang-Qian;  Chen, Xue-Chun;  Luo, Jiao;  Li, Chao;  Wang, Yi;  Shi, Da-Yong
Adobe PDF(824Kb)  |  收藏  |  浏览/下载:285/0  |  提交时间:2019/08/21
Pyrimidinedionederivatives  DPP-4 inhibitor  Molecular hybrid  SARs  Type 2 diabetes  
新型氟代PTP1B抑制剂的设计、合成及活性研究 学位论文
, 北京: 中国科学院大学, 2016
作者:  王保程
Adobe PDF(4845Kb)  |  收藏  |  浏览/下载:261/0  |  提交时间:2016/05/31
糖尿病  氟代化合物  Ptp1b抑制剂  计算机辅助药物设计  分子对接  
Halogenated Organic Molecules of Rhodomelaceae Origin: Chemistry and Biology 期刊论文
CHEMICAL REVIEWS, 2013, 卷号: 113, 期号: 5, 页码: 3632-3685
作者:  Wang, Bin-Gui;  Gloer, James B.;  Ji, Nai-Yun;  Zhao, Jian-Chun;  Wang, BG
Adobe PDF(9186Kb)  |  收藏  |  浏览/下载:297/0  |  提交时间:2014/07/17
Synthesis of three bromophenols from red algae as PTP1B inhibitors 期刊论文
CHINESE JOURNAL OF OCEANOLOGY AND LIMNOLOGY, 2011, 卷号: 29, 期号: 1, 页码: 68-74
作者:  Guo Shuju;  Li Jing;  Li Ting;  Shi Dayong;  Han Lijun
Adobe PDF(360Kb)  |  收藏  |  浏览/下载:373/0  |  提交时间:2012/07/03
Bromophenols  Synthesis  Ptp1b Inhibitory Activity