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Palladium-Catalyzed Remote C-H Phosphonylation of Indoles at the C4 and C6 Positions by a Radical Approach 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 7
作者:  Shi, Xiaolin;  Wang, Zemin;  Li, Yuxiu;  Li, Xiaowei;  Li, Xiangqian;  Shi, Dayong
Adobe PDF(1762Kb)  |  收藏  |  浏览/下载:194/0  |  提交时间:2021/06/04
C−  H activation  indoles  palladium  phosphonylation  regioselectivity  
Antidiabetic activity in vitro and in vivo of BDB, a selective inhibitor of protein tyrosine phosphatase 1B, fromRhodomela confervoides 期刊论文
BRITISH JOURNAL OF PHARMACOLOGY, 2020, 卷号: 177, 期号: 19, 页码: 4464-4480
作者:  Luo, Jiao;  Zheng, Meiling;  Jiang, Bo;  Li, Chao;  Guo, Shuju;  Wang, Lijun;  Li, Xiangqian;  Yu, Rilei;  Shi, Dayong
Adobe PDF(42653Kb)  |  收藏  |  浏览/下载:287/0  |  提交时间:2020/09/29
bromophenol  PTP1B inhibitor  selectivity  cell permeability  oral bioavailability  
AcOH-mediated aerobic oxidative synthesis of 2-thioalkylbenzothiazoles via a three-component reaction 期刊论文
TETRAHEDRON LETTERS, 2020, 卷号: 61, 期号: 26, 页码: 5
作者:  Li, Xiaowei;  Li, Yuxiu;  Liu, Ruihua;  Wang, Zemin;  Li, Xiangqian;  Shi, Dayong
Adobe PDF(819Kb)  |  收藏  |  浏览/下载:152/0  |  提交时间:2020/09/25
2-Thioalkylbenzothiazoles  Metal-free  Aerobic oxidation  Multicomponent reaction  
Structural and Bioactive Studies of Halogenated Constituents from Sponges 期刊论文
CURRENT MEDICINAL CHEMISTRY, 2020, 卷号: 27, 期号: 14, 页码: 2335-2360
作者:  Li, Chao;  Shi, Dayong
收藏  |  浏览/下载:200/0  |  提交时间:2020/09/24
Halogenated  sponges  marine  isolate  constitutes  activity  
Inhibition of PTP1B blocks pancreatic cancer progression by targeting the PKM2/AMPK/mTOC1 pathway 期刊论文
CELL DEATH & DISEASE, 2019, 卷号: 10, 页码: 15
作者:  Xu, Qi;  Wu, Ning;  Li, Xiangqian;  Guo, Chuanlong;  Li, Chao;  Jiang, Bo;  Wang, Huaizhi;  Shi, Dayong
Adobe PDF(3632Kb)  |  收藏  |  浏览/下载:285/0  |  提交时间:2020/03/20
Recent advances in transition-metal-catalyzed incorporation of fluorine-containing groups 期刊论文
BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 15, 页码: 2213-2270
作者:  Li, Xiaowei;  Shi, Xiaolin;  Li, Xiangqian;  Shi, Dayong
Adobe PDF(5059Kb)  |  收藏  |  浏览/下载:262/0  |  提交时间:2020/01/03
catalysis  C-R-F bond  fluorination  fluoroalkylation  transition metals  
Ligand- and Additive-Free 2-Position-Selective Trifluoromethylation of Heteroarenes Under Ambient Conditions 期刊论文
FRONTIERS IN CHEMISTRY, 2019, 卷号: 7, 页码: 10
作者:  Shi, Xiaolin;  Li, Xiaowei;  Li, Xiangqian;  Shi, Dayong
Adobe PDF(988Kb)  |  收藏  |  浏览/下载:254/0  |  提交时间:2020/01/03
C-H functionalization  trifluoromethylation  indoles  copper  radical reaction  
Design, synthesis and biological evaluation of bromophenol-thiazolylhydrazone hybrids inhibiting the interaction of translation initiation factors eIF4E/eIF4G as multifunctional agents for cancer treatment 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 177, 页码: 153-170
作者:  Wang, Lijun;  Guo, Chuanlong;  Li, Xiuxue;  Yu, Xuemin;  Li, Xiangqian;  Xu, Kuo;  Jiang, Bo;  Jia, Xiaoling;  Li, Chao;  Shi, Dayong
Adobe PDF(4835Kb)  |  收藏  |  浏览/下载:321/0  |  提交时间:2019/08/29
Bromophenol-thiazolylhydrazone hybrids  Synthesis  Multifunctional agents  eIF4E/eIF4G interaction  Autophagy  ROS  
Chalcone-analogue fluorescent probes for detecting thiophenols in seawater samples 期刊论文
TALANTA, 2019, 卷号: 201, 页码: 301-308
作者:  Liu, Hua;  Guo, Chuanlong;  Guo, Shuju;  Fan, Junting;  Wang, Lijun;  Shi, Dayong
Adobe PDF(1820Kb)  |  收藏  |  浏览/下载:273/0  |  提交时间:2019/08/29
Fluorescent probe  Thiophenol  Seawater sample  Chalcone  
Highly Selective Protein Tyrosine Phosphatase Inhibitor, 2,2 ',3,3 '-Tetrabromo-4,4 ',5,5 '-tetrahydroxydiphenylmethane, Ameliorates Type 2 Diabetes Mellitus in BKS db Mice 期刊论文
MOLECULAR PHARMACEUTICS, 2019, 卷号: 16, 期号: 5, 页码: 1839-1850
作者:  Li, Chao;  Luo, Jiao;  Guo, Shuju;  Jia, Xiaoling;  Guo, Chuanlong;  Li, Xiangqian;  Xu, Qi;  Shi, Dayong
收藏  |  浏览/下载:309/0  |  提交时间:2019/08/28
type 2 diabetes mellitus  protein tyrosine phosphatase 1B  insulin resistance  hypoglycemic activity  dyslipidemia