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Palladium-Catalyzed Remote C-H Phosphonylation of Indoles at the C4 and C6 Positions by a Radical Approach 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 7
作者:  Shi, Xiaolin;  Wang, Zemin;  Li, Yuxiu;  Li, Xiaowei;  Li, Xiangqian;  Shi, Dayong
Adobe PDF(1762Kb)  |  收藏  |  浏览/下载:194/0  |  提交时间:2021/06/04
C−  H activation  indoles  palladium  phosphonylation  regioselectivity  
Antidiabetic activity in vitro and in vivo of BDB, a selective inhibitor of protein tyrosine phosphatase 1B, fromRhodomela confervoides 期刊论文
BRITISH JOURNAL OF PHARMACOLOGY, 2020, 卷号: 177, 期号: 19, 页码: 4464-4480
作者:  Luo, Jiao;  Zheng, Meiling;  Jiang, Bo;  Li, Chao;  Guo, Shuju;  Wang, Lijun;  Li, Xiangqian;  Yu, Rilei;  Shi, Dayong
Adobe PDF(42653Kb)  |  收藏  |  浏览/下载:288/0  |  提交时间:2020/09/29
bromophenol  PTP1B inhibitor  selectivity  cell permeability  oral bioavailability  
AcOH-mediated aerobic oxidative synthesis of 2-thioalkylbenzothiazoles via a three-component reaction 期刊论文
TETRAHEDRON LETTERS, 2020, 卷号: 61, 期号: 26, 页码: 5
作者:  Li, Xiaowei;  Li, Yuxiu;  Liu, Ruihua;  Wang, Zemin;  Li, Xiangqian;  Shi, Dayong
Adobe PDF(819Kb)  |  收藏  |  浏览/下载:152/0  |  提交时间:2020/09/25
2-Thioalkylbenzothiazoles  Metal-free  Aerobic oxidation  Multicomponent reaction  
An UHPLC-TOF-MS method for quantifying novel brominated anticancer compound bromophenol-thiosemicarbazone hybrid and its application to in vivo pharmacokinetic study 期刊论文
JOURNAL OF ANALYTICAL SCIENCE AND TECHNOLOGY, 2020, 卷号: 11, 期号: 1, 页码: 7
作者:  Li, Xiuxue;  Wang, Lijun;  Jia, Xiaoling;  Guo, Chuanlong;  Li, Chao;  Zhang, Jiajia;  Shi, Dayong
Adobe PDF(579Kb)  |  收藏  |  浏览/下载:155/0  |  提交时间:2020/09/23
Novel compound  Quantitation  UHPLC-TOF-MS  Pharmacokinetics  
Inhibition of PTP1B blocks pancreatic cancer progression by targeting the PKM2/AMPK/mTOC1 pathway 期刊论文
CELL DEATH & DISEASE, 2019, 卷号: 10, 页码: 15
作者:  Xu, Qi;  Wu, Ning;  Li, Xiangqian;  Guo, Chuanlong;  Li, Chao;  Jiang, Bo;  Wang, Huaizhi;  Shi, Dayong
Adobe PDF(3632Kb)  |  收藏  |  浏览/下载:286/0  |  提交时间:2020/03/20
Design, synthesis and biological evaluation of bromophenol-thiazolylhydrazone hybrids inhibiting the interaction of translation initiation factors eIF4E/eIF4G as multifunctional agents for cancer treatment 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 177, 页码: 153-170
作者:  Wang, Lijun;  Guo, Chuanlong;  Li, Xiuxue;  Yu, Xuemin;  Li, Xiangqian;  Xu, Kuo;  Jiang, Bo;  Jia, Xiaoling;  Li, Chao;  Shi, Dayong
Adobe PDF(4835Kb)  |  收藏  |  浏览/下载:321/0  |  提交时间:2019/08/29
Bromophenol-thiazolylhydrazone hybrids  Synthesis  Multifunctional agents  eIF4E/eIF4G interaction  Autophagy  ROS  
Chalcone-analogue fluorescent probes for detecting thiophenols in seawater samples 期刊论文
TALANTA, 2019, 卷号: 201, 页码: 301-308
作者:  Liu, Hua;  Guo, Chuanlong;  Guo, Shuju;  Fan, Junting;  Wang, Lijun;  Shi, Dayong
Adobe PDF(1820Kb)  |  收藏  |  浏览/下载:273/0  |  提交时间:2019/08/29
Fluorescent probe  Thiophenol  Seawater sample  Chalcone  
BOS-93, a novel bromophenol derivative, induces apoptosis and autophagy in human A549 lung cancer cells via PI3K/Akt/mTOR and MAPK signaling pathway 期刊论文
EXPERIMENTAL AND THERAPEUTIC MEDICINE, 2019, 卷号: 17, 期号: 5, 页码: 3848-3858
作者:  Guo, Chuanlong;  Wang, Lijun;  Zhao, Yue;  Jiang, Bo;  Luo, Jiao;  Shi, Dayong
Adobe PDF(2683Kb)  |  收藏  |  浏览/下载:235/0  |  提交时间:2019/08/28
bromophenol  apoptosis  autophagy  phosphoinositide 3-kinase  protein kinase B  mechanistic target of rapamycin signaling  reactive oxygen species  
Design and Synthesis of a Fluorescent Probe with a Large Stokes Shift for Detecting Thiophenols and Its Application in Water Samples and Living Cells 期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 2, 页码: 14
作者:  Liu, Hua;  Guo, Chuanlong;  Guo, Shuju;  Wang, Lijun;  Shi, Dayong
Adobe PDF(2843Kb)  |  收藏  |  浏览/下载:255/0  |  提交时间:2019/08/27
fluorescent probe  thiophenol  water samples  chalcone  living cells  
Bromophenol curcumin analog BCA-5 exerts an antiangiogenic effect through the HIF-1 alpha/VEGF/Akt signaling pathway in human umbilical vein endothelial cells 期刊论文
ANTI-CANCER DRUGS, 2018, 卷号: 29, 期号: 10, 页码: 965-974
作者:  Guo, Chuanlong;  Wang, Lijun;  Jiang, Bo;  Shi, Dayong
收藏  |  浏览/下载:228/0  |  提交时间:2019/05/15
antiangiogenesis  curcumin analogs  hypoxia-inducible factor-1 alpha  human umbilical vein endothelial cells  vascular endothelial growth factor