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中国科学院海洋研究所机构知识库
Knowledge Management System Of Institute of Oceanology, Chinese Academy of Sciences
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EGPI-1, a novel eIF4E/eIF4G interaction inhibitor, inhibits lung cancer cell growth and angiogenesis through Ras/MNK/ERK/eIF4E signaling pathway
期刊论文
CHEMICO-BIOLOGICAL INTERACTIONS, 2022, 卷号: 352, 页码: 10
作者:
Qi, Xueju
;
Zhang, Shuna
;
Chen, Zekun
;
Wang, Lijun
;
Zhu, Wenyong
;
Yin, Chuanjin
;
Fan, Junting
;
Wu, Xiaochen
;
Wang, Jing
;
Guo, Chuanlong
Adobe PDF(10635Kb)
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浏览/下载:112/0
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提交时间:2022/07/18
Human lung cancer
eIF4E
EGPI-1
Anticancer
Angiogenesis
Naturally occurring ureidobromophenols with potent antioxidant activities from the marine red alga Rhodomela confervoides
期刊论文
ALGAL RESEARCH-BIOMASS BIOFUELS AND BIOPRODUCTS, 2021, 卷号: 56, 页码: 5
作者:
Li, Ke
;
Li, Xiao-Ming
;
Gloer, James B.
;
Wang, Bin-Gui
Adobe PDF(541Kb)
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浏览/下载:127/0
  |  
提交时间:2021/12/07
Marine red alga
Rhodomela confervoides
Ureidobromophenols
Antioxidant activity
Discovery of 5-(3-bromo-2-(2,3-dibromo-4,5-dimethoxybenzyl)-4,5-dimethoxybenzylidene)thiazolidine-2,4-dione as a novel potent protein tyrosine phosphatase 1B inhibitor with antidiabetic properties
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 108, 页码: 13
作者:
Jiang, Bo
;
Luo, Jiao
;
Guo, Shuju
;
Wang, Lijun
Adobe PDF(8153Kb)
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浏览/下载:181/0
  |  
提交时间:2021/05/11
Type 2 diabetes mellitus
Protein tyrosine phosphatase 1B inhibitors
Thiazolidinedione
Insulin signaling
Anti-diabetic activities
First Succinylome Profiling of Vibrio alginolyticus Reveals Key Role of Lysine Succinylation in Cellular Metabolism and Virulence
期刊论文
FRONTIERS IN CELLULAR AND INFECTION MICROBIOLOGY, 2021, 卷号: 10, 页码: 13
作者:
Zeng, Fuyuan
;
Pang, Huanying
;
Chen, Ying
;
Zheng, Hongwei
;
Li, Wanxin
;
Ramanathan, Srinivasan
;
Hoare, Rowena
;
Monaghan, Sean J.
;
Lin, Xiangmin
;
Jian, Jichang
Adobe PDF(2471Kb)
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浏览/下载:191/0
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提交时间:2021/04/14
Vibrio alginolyticus
lysine succinylation
acetylation
crosstalk
virulence factors
Investigating the properties of nano core-shell CeO2@C as haloperoxidase mimicry catalyst for antifouling applications
期刊论文
COLLOIDS AND SURFACES A-PHYSICOCHEMICAL AND ENGINEERING ASPECTS, 2021, 卷号: 608, 页码: 9
作者:
Wang, Nan
;
Li, Wangqiang
;
Ren, Yadong
;
Duan, Jizhou
;
Zhai, Xiaofan
;
Guan, Fang
;
Wang, Lifei
;
Hou, Baorong
Adobe PDF(6587Kb)
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浏览/下载:181/0
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提交时间:2021/04/12
CeO2@C
Haloperoxidase mimicry catalyst
Haloperoxidase-like activity
Hypobromous acid
Antibacterial activity
Antifouling
Characterization and function analysis of a Kazal-type serine proteinase inhibitor in the red claw crayfish Cherax quadricarinatus
期刊论文
DEVELOPMENTAL AND COMPARATIVE IMMUNOLOGY, 2021, 卷号: 114, 页码: 10
作者:
Wang, Yan
;
Wang, Baojie
;
Liu, Mei
;
Jiang, Keyong
;
Wang, Mengqiang
;
Wang, Lei
Adobe PDF(5359Kb)
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浏览/下载:178/0
  |  
提交时间:2021/04/12
Cherax quadricarinatus
Kazal-type serine proteinase inhibitor
Innate immunity
Novel poly (ADP-ribose) polymerases inhibitor DHC-1 exhibits in vitro and in vivo anticancer activity on BRCA-deficient pancreatic cancer cells
期刊论文
FOOD AND CHEMICAL TOXICOLOGY, 2021, 卷号: 147, 页码: 10
作者:
Wu, Xiaochen
;
Li, Qiqi
;
Zhang, Fan
;
Wang, Lijun
;
Wang, Jun
;
Fan, Junting
;
Di, Guohu
;
Guo, Chuanlong
Adobe PDF(8144Kb)
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收藏
  |  
浏览/下载:166/0
  |  
提交时间:2021/04/21
PARP inhibitor
BRCA
Pancreatic cancer
Binding properties of marine bromophenols with human protein tyrosine phosphatase 1B: Molecular docking, surface plasmon resonance and cellular insulin resistance study
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2020, 卷号: 163, 页码: 200-208
作者:
Luo, Jiao
;
Zhang, Renshuai
;
Wang, Xuehe
;
Hou, Zhanhui
;
Guo, Shuju
;
Jiang, Bo
Adobe PDF(3013Kb)
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  |  
浏览/下载:152/0
  |  
提交时间:2021/04/12
PTP1B
Bromophenol
Molecular docking
Surface plasmon resonance
Antidiabetic activity in vitro and in vivo of BDB, a selective inhibitor of protein tyrosine phosphatase 1B, fromRhodomela confervoides
期刊论文
BRITISH JOURNAL OF PHARMACOLOGY, 2020, 卷号: 177, 期号: 19, 页码: 4464-4480
作者:
Luo, Jiao
;
Zheng, Meiling
;
Jiang, Bo
;
Li, Chao
;
Guo, Shuju
;
Wang, Lijun
;
Li, Xiangqian
;
Yu, Rilei
;
Shi, Dayong
Adobe PDF(42653Kb)
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浏览/下载:263/0
  |  
提交时间:2020/09/29
bromophenol
PTP1B inhibitor
selectivity
cell permeability
oral bioavailability
Novel eIF4E/eIF4G protein-protein interaction inhibitors DDH-1 exhibits anti-cancer activity in vivo and in vitro
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2020, 卷号: 160, 页码: 496-505
作者:
Wang, Jun
;
Wang, Lijun
;
Zhang, Shuhong
;
Fan, Junting
;
Yang, Hui
;
Li, Qiqi
;
Guo, Chuanlong
Adobe PDF(3920Kb)
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收藏
  |  
浏览/下载:179/0
  |  
提交时间:2020/10/26
eIF4E/eIF4G
Human lung cancer
Apoptosis
DNA damage
ROS