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中国科学院海洋研究所机构知识库
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Design of Chitosan Sterilization Agents by a Structure Combination Strategy and Their Potential Application in Crop Protection
期刊论文
MOLECULES, 2021, 卷号: 26, 期号: 11, 页码: 15
作者:
Liu, Weixiang
;
Qin, Yukun
;
Li, Pengcheng
Adobe PDF(1133Kb)
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浏览/下载:131/0
  |  
提交时间:2021/12/07
chitosan derivative
structure combination strategy
modification
agriculture
antimicrobial application
Novel poly (ADP-ribose) polymerases inhibitor DHC-1 exhibits in vitro and in vivo anticancer activity on BRCA-deficient pancreatic cancer cells
期刊论文
FOOD AND CHEMICAL TOXICOLOGY, 2021, 卷号: 147, 页码: 10
作者:
Wu, Xiaochen
;
Li, Qiqi
;
Zhang, Fan
;
Wang, Lijun
;
Wang, Jun
;
Fan, Junting
;
Di, Guohu
;
Guo, Chuanlong
Adobe PDF(8144Kb)
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浏览/下载:166/0
  |  
提交时间:2021/04/21
PARP inhibitor
BRCA
Pancreatic cancer
BTH-8, a novel poly (ADP-ribose) polymerase-1 (PARP-1) inhibitor, causes DNA double-strand breaks and exhibits anticancer activities in vitro and in vivo
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2020, 卷号: 150, 页码: 238-245
作者:
Guo, Chuanlong
;
Zhang, Fan
;
Wu, Xiaochen
;
Yu, Xuemin
;
Wu, Xianggen
;
Shi, Dayong
;
Wang, Lijun
Adobe PDF(1767Kb)
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浏览/下载:155/0
  |  
提交时间:2020/09/23
PARP-1 inhibitor
DNA double-strand breaks
HCC-1937
In vivo
Apoptosis
An UHPLC-TOF-MS method for quantifying novel brominated anticancer compound bromophenol-thiosemicarbazone hybrid and its application to in vivo pharmacokinetic study
期刊论文
JOURNAL OF ANALYTICAL SCIENCE AND TECHNOLOGY, 2020, 卷号: 11, 期号: 1, 页码: 7
作者:
Li, Xiuxue
;
Wang, Lijun
;
Jia, Xiaoling
;
Guo, Chuanlong
;
Li, Chao
;
Zhang, Jiajia
;
Shi, Dayong
Adobe PDF(579Kb)
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浏览/下载:141/0
  |  
提交时间:2020/09/23
Novel compound
Quantitation
UHPLC-TOF-MS
Pharmacokinetics
Superamphiphobic aluminum alloy with low sliding angles and acid-alkali liquids repellency
期刊论文
MATERIALS & DESIGN, 2020, 卷号: 188, 页码: 9
作者:
Zhang, Binbin
;
Zeng, Yuxiang
;
Wang, Jia
;
Sun, Yuanyuan
;
Zhang, Jie
;
Li, Yantao
Adobe PDF(4036Kb)
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浏览/下载:152/0
  |  
提交时间:2020/09/23
Micro-nano
Superhydrophobic
Superamphiphobic
Chemical stability
Self-cleaning
The Fluoro-Thiazolylhydrazone Compound TSC-3C Inhibits Triple Negative Breast Cancer (TNBC) Cell Line Activity by Promoting Apoptosis, Regulating the MAPK Pathway and Inducing Mitochondrial Dysfunction
期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2020, 卷号: 21, 期号: 3, 页码: 15
作者:
Zhang, Jiajia
;
Dai, Jiajia
;
Zheng, Qingxuan
;
Guo, Shuju
;
Yu, Yanyan
;
Hu, Wenpeng
;
Gao, Yanan
;
Shi, Dayong
Adobe PDF(2858Kb)
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浏览/下载:132/0
  |  
提交时间:2020/09/23
triple negative breast cancer
MDA-MB-231 cells
fluoro-thiazolylhydrazone
MAPK pathway
phosphorylated p44/42 MAPK (ERK1/2)
phosphorylated c-Jun N-terminal kinase (p-JNK)
apoptosis
Design, synthesis and biological evaluation of bromophenol-thiazolylhydrazone hybrids inhibiting the interaction of translation initiation factors eIF4E/eIF4G as multifunctional agents for cancer treatment
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 177, 页码: 153-170
作者:
Wang, Lijun
;
Guo, Chuanlong
;
Li, Xiuxue
;
Yu, Xuemin
;
Li, Xiangqian
;
Xu, Kuo
;
Jiang, Bo
;
Jia, Xiaoling
;
Li, Chao
;
Shi, Dayong
Adobe PDF(4835Kb)
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  |  
浏览/下载:294/0
  |  
提交时间:2019/08/29
Bromophenol-thiazolylhydrazone hybrids
Synthesis
Multifunctional agents
eIF4E/eIF4G interaction
Autophagy
ROS
Discovery of Novel Bromophenol Thiosemicarbazone Hybrids as Potent Selective Inhibitors of Poly(ADP-ribose) Polymerase-1 (PARP-1) for Use in Cancer
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 6, 页码: 3051-3067
作者:
Guo, Chuanlong
;
Wang, Lijun
;
Li, Xinxue
;
Wang, Shuaiyu
;
Yu, Xuemin
;
Xu, Kuo
;
Zhao, Yue
;
Luo, Jiao
;
Li, Xiangqian
;
Jiang, Bo
;
Shi, Dayong
Adobe PDF(8824Kb)
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  |  
浏览/下载:299/0
  |  
提交时间:2019/08/28
Cyclization Reaction of Acyl Thiourea Chitosan: Enhanced Antifungal Properties via Structural Optimization
期刊论文
MOLECULES, 2018, 卷号: 23, 期号: 3, 页码: 13
作者:
Qin, Yukun
;
Liu, Weixiang
;
Xing, Ronge
;
Liu, Song
;
Li, Kecheng
;
Li, Pengcheng
Adobe PDF(5247Kb)
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  |  
浏览/下载:217/0
  |  
提交时间:2019/08/21
synthesis
1,2,4-triazolyl
acyl thiourea
chitosan
antifungal activity
A novel fluorinated thiosemicarbazone derivative-2-(3,4-difluorobenzylidene) hydrazinecarbothioamide induces apoptosis in human A549 lung cancer cells via ROS-mediated mitochondria-dependent pathway
期刊论文
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2017, 卷号: 491, 期号: 1, 页码: 65-71
作者:
Zhao, Yue
;
Guo, Chuanlong
;
Wang, Lijun
;
Wang, Shuaiyu
;
Li, Xiangqian
;
Jiang, Bo
;
Wu, Ning
;
Guo, Shuju
;
Zhang, Renshuai
;
Liu, Kun
;
Shi, Dayong
Adobe PDF(1849Kb)
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收藏
  |  
浏览/下载:320/0
  |  
提交时间:2018/01/11
Thiosemicarbazone
Anticancer
2-(3
Apoptosis
4-difluorobenzylidene) Hydrazinecarbothioamide
Ros
Mitochondria-dependent Pathway